N-heterocyclic carbene switchable radical or benzyne meditated arylation of thiols using DMF/KOtBu

Title
N-heterocyclic carbene switchable radical or benzyne meditated arylation of thiols using DMF/KOtBu
Publication Date
2025
Author(s)
Puschnig, Johannes
Greatrex, Ben W
( author )
OrcID: https://orcid.org/0000-0002-0356-4966
Email: bgreatre@une.edu.au
UNE Id une-id:bgreatre
Type of document
Journal Article
Language
en
Entity Type
Publication
Publisher
Georg Thieme Verlag
Place of publication
Germany
DOI
10.1055/a-2460-8302
UNE publication id
une:1959.11/63846
Abstract

A mild, metal and photoredox-free direct arylation of alkyl and aryl thiols with aryl iodides using a DMF/KOtBu system has been developed. In the absence of an N-heterocyclic carbene (NHC) additive, the reaction proceeds via a benzyne intermediate and was suitable for the substitution of thiols with phenyl, while the presence of an NHC or phenanthroline derivative improves regioselectivity for the reaction of substituted aryl iodides via a radical pathway. This protocol features inexpensive materials and good substrate scope, and could be useful in the arylation of aryl and alkyl thiols.

Link
Citation
Synlett, 36(7), p. 884-888
Start page
884
End page
888

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