| Author(s) |
Wilkinson, Brendan
|
| Publication Date |
2013
|
| Abstract |
Acylated derivatives of 1-hydroxybenzotriazole (HOBt) have been widely used as reactive intermediates in a variety of one-pot, bond forming reactions. Isolable benzotriazole 'esters' 1-(benzoyloxy)benzotriazole (1-BBTZ, 1) and 1-(acetoxy)benzotriazole (2) are also useful reagents for the regioselective acylation of diols and partially protected carbohydrates (Fig. 1).[¹] 1-(Acyloxy) benzotriazoles 1 and 2 can be conveniently prepared by a carbodiimide-promoted condensation of HOBt,[²] or via the corresponding acyl chloride.[¹]
|
| Citation |
Australian Journal of Chemistry, 66(8), p. 910-912
|
| ISSN |
1445-0038
0004-9425
|
| Link | |
| Language |
en
|
| Publisher |
CSIRO Publishing
|
| Title |
1-(Acyloxy)benzotriazoles: Useful Reagents for the Regioselective Acylation of Diols
|
| Type of document |
Journal Article
|
| Entity Type |
Publication
|
| Name | Size | format | Description | Link |
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